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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $941 | In Stock | |
5 mg | $1,880 | In Stock | |
10 mg | $2,560 | In Stock | |
25 mg | $3,780 | In Stock | |
50 mg | $5,130 | In Stock | |
100 mg | $6,920 | In Stock | |
1 mL x 10 mM (in DMSO) | $3,910 | In Stock |
Description | AR-M 1896 Acetate is the selective agonist of GalR2. |
In vitro | Removal of the glycine residue in position 1 resulted in AR-M1896 with almost unchanged GalR2 affinity and functional activity, and 500-fold selectivity for GalR2-Rs over GalR1-Rs[1].? |
In vivo | In normal rats mechanical and cold allodynia of the hindpaw are induced by intrathecal infusion of low-dose galanin. The same effect is seen with equimolar doses of AR-M1896 or AR-M961 (an agonist both at GalR1 and GalR2 receptors). In allodynic Bennett model rats, the mechanical threshold dose-dependently increased after intrathecal injection of a high AR-M961dose, whereas no effect was observed in the control or AR-M1896 group. No effect of either compounds was observed in nonallodynic Bennett model rats[1]. |
Alias | AR-M 1896 Acetate (367518-31-8 Free base) |
Molecular Weight | 1196.35 |
Formula | C56H85N13O16 |
Cas No. |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | |||||||||||||||||||||||||
Solubility Information | DMSO: 55 mg/ml (45.97 mM) ![]() | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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